PREPARATION OF 3-AMINO-1,4-BENZODIAZEPIN-2-ONES VIA DIRECT AZIDATION WITH TRISYL AZIDE

Authors
BUTCHER JW LIVERTON NJ SELNICK HG ELLIOT JM SMITH GR TEBBEN AJ PRIBUSH DA WAI JS CLAREMON DA
Citation
Jw. Butcher et al., PREPARATION OF 3-AMINO-1,4-BENZODIAZEPIN-2-ONES VIA DIRECT AZIDATION WITH TRISYL AZIDE, Tetrahedron letters, 37(37), 1996, pp. 6685-6688
Citations number
13
Categorie Soggetti
Chemistry Inorganic & Nuclear
Journal title
Tetrahedron letters → ACNP
ISSN journal
00404039
Volume
37
Issue
37
Year of publication
1996
Pages
6685 - 6688
Database
ISI
SICI code
0040-4039(1996)37:37<6685:PO3VDA>2.0.ZU;2-F
Abstract
An efficient synthesis of 3-amino-1,4-benzodiazepin-2-ones utilizing t riisopropylbenzenesulfonyl azide (trisyl azide) for the direct azidati on of 1,4-benzodiazepin-2-ones is described. Copyright (C) 1996 Elsevi er Science Ltd