A SYNTHESIS OF FUNCTIONALIZED INDOLINE 2,2-BISCARBOXYLATES

Authors
WRIGHT SW DOW RL MCCLURE LD HAGEMAN DL
Citation
Sw. Wright et al., A SYNTHESIS OF FUNCTIONALIZED INDOLINE 2,2-BISCARBOXYLATES, Tetrahedron letters, 37(39), 1996, pp. 6965-6968
Citations number
12
Categorie Soggetti
Chemistry Inorganic & Nuclear
Journal title
Tetrahedron letters → ACNP
ISSN journal
00404039
Volume
37
Issue
39
Year of publication
1996
Pages
6965 - 6968
Database
ISI
SICI code
0040-4039(1996)37:39<6965:ASOFI2>2.0.ZU;2-O
Abstract
A synthetic approach to a structurally novel series of indoline 2,2-bi scarboxylates is employs a tandem bis-alkylation strategy to cyclize t he indoline heteroring from the bromide 7 and diethyl bromomalonate. T he indolines thus prepared may be N-deprotected and further functional ized on the indoline nitrogen. Copyright (C) 1996 Elsevier Science Ltd