SYNTHESIS OF YL(2R,3R)-2-CYANO-3-FORMYL-AZIRIDINE-1-CARBOXYLATE - A NEW POTENTIAL BUILDING-BLOCK FOR AMINO-ALCOHOLS AND POLYAMINES

Authors
JAHNISCH K
Citation
K. Jahnisch, SYNTHESIS OF YL(2R,3R)-2-CYANO-3-FORMYL-AZIRIDINE-1-CARBOXYLATE - A NEW POTENTIAL BUILDING-BLOCK FOR AMINO-ALCOHOLS AND POLYAMINES, Tetrahedron letters, 38(2), 1997, pp. 227-228
Citations number
4
Categorie Soggetti
Chemistry Inorganic & Nuclear
Journal title
Tetrahedron letters → ACNP
ISSN journal
00404039
Volume
38
Issue
2
Year of publication
1997
Pages
227 - 228
Database
ISI
SICI code
0040-4039(1997)38:2<227:SOY-AN>2.0.ZU;2-P
Abstract
The cyano dihydroxyethyl aziridine 3 was obtained by acid catalyzed hy drolysis of the acetonide protected aziridine 2. Subsequent transforma tion by glycol cleavage yielded tert-butyl (2R,3R)-2-cyano-3-formyl-az iri-dine-1-carboxylate (4). Copyright (C) 1996 Elsevier Science Ltd