SYNTHESIS OF N-PROTECTED GAMMA-AMINO-BETA-KETO-ESTERS FROM URETHANE N-CARBOXYANHYDRIDES (UNCAS)

Authors
PARIS M FEHRENTZ JA HEITZ A LOFFET A MARTINEZ J
Citation
M. Paris et al., SYNTHESIS OF N-PROTECTED GAMMA-AMINO-BETA-KETO-ESTERS FROM URETHANE N-CARBOXYANHYDRIDES (UNCAS), Tetrahedron letters, 37(47), 1996, pp. 8489-8492
Citations number
14
Categorie Soggetti
Chemistry Inorganic & Nuclear
Journal title
Tetrahedron letters → ACNP
ISSN journal
00404039
Volume
37
Issue
47
Year of publication
1996
Pages
8489 - 8492
Database
ISI
SICI code
0040-4039(1996)37:47<8489:SONGFU>2.0.ZU;2-3
Abstract
N-protected gamma-amino-beta-keto-esters were synthesized from the cor responding N-protected N-carboxyanhydride (UNCAs) by reaction with the lithium enolate of ethyl acetate in good yields. These compounds are precursors of statine derivatives. Copyright (C) 1996 Elsevier Science Ltd