SYNTHESIS OF C-14-LABELED LEVAMISOLE AND C-13-LABELED TETRAMISOLE

Authors
Citation
Vj. Feil, SYNTHESIS OF C-14-LABELED LEVAMISOLE AND C-13-LABELED TETRAMISOLE, Journal of labelled compounds & radiopharmaceuticals, 38(12), 1996, pp. 1071-1076
Citations number
7
Categorie Soggetti
Chemistry Analytical","Pharmacology & Pharmacy","Biochemical Research Methods
ISSN journal
03624803
Volume
38
Issue
12
Year of publication
1996
Pages
1071 - 1076
Database
ISI
SICI code
0362-4803(1996)38:12<1071:SOCLAC>2.0.ZU;2-R
Abstract
The syntheses of C-14-ring labeled levamisole 2,3,5,6-tetrahydro-6-phe nyl[C-14-UL]imidazo[2,1-b] thiazole) from acetophenone-ring-UL-C-14 in 5 steps plus resolution with a 7.5% overall yield, and C-13(6)-ring l abeled tetramisole 2,3,5,6-tetrahydro-6-phenyl[C-13(6)]imidazo[2,1-b] thiazole) from benzene-C-13(6) in 6 steps with a 9.0% overall yield ar e described.