A VERSATILE SYNTHESIS OF 3-SUBSTITUTED INDOLES

Authors
KATRITZKY AR XIE LH CUNDY D
Citation
Ar. Katritzky et al., A VERSATILE SYNTHESIS OF 3-SUBSTITUTED INDOLES, Synthetic communications, 25(4), 1995, pp. 539-551
Citations number
17
Categorie Soggetti
Chemistry Inorganic & Nuclear
Journal title
Synthetic communications → ACNP
ISSN journal
00397911
Volume
25
Issue
4
Year of publication
1995
Pages
539 - 551
Database
ISI
SICI code
0039-7911(1995)25:4<539:AVSO3I>2.0.ZU;2-L
Abstract
A variety of 3-substituted indoles are prepared from 1-methyl-3-(benzo triazol-1-ylalkyl)indoles (1), which are readily available either from the condensation of 3-methylindole with N-(benzotriazol-1-ylalkyl)car bamates or from the alkylation and silylation of lithiated 1-methyl-3- (benzotriazol-1-ylmethyl)indole (2).