ASYMMETRIC-SYNTHESIS .36. SYNTHESIS OF TETRAHYDROAZOCINES BY [2-DIHYDROPYRIDINE(2] THERMAL CYCLOADDITION TO LATENT 1,4)

Authors
LALLEMAND MC CHIADMI M TOMAS A KUNESCH N HUSSON HP
Citation
Mc. Lallemand et al., ASYMMETRIC-SYNTHESIS .36. SYNTHESIS OF TETRAHYDROAZOCINES BY [2-DIHYDROPYRIDINE(2] THERMAL CYCLOADDITION TO LATENT 1,4), Tetrahedron letters, 36(12), 1995, pp. 2053-2056
Citations number
20
Categorie Soggetti
Chemistry Inorganic & Nuclear
Journal title
Tetrahedron letters → ACNP
ISSN journal
00404039
Volume
36
Issue
12
Year of publication
1995
Pages
2053 - 2056
Database
ISI
SICI code
0040-4039(1995)36:12<2053:A.SOTB>2.0.ZU;2-L
Abstract
The regiospecific formation of tetrahydroazocines 7-9 by [2+2] cycload dition of an activated alkyne to substrates of type 1 is reported. Thi s procedure provides a simple access to chiral functionalized eight-me mbered rings.