THE STEREOSPECIFIC SYNTHESIS OF (2S,3R) 3-CARBOXYPROLINE AND (2S,3R) 3-AMINOPROLINE

Authors
BALDWIN JE ADLINGTON RM GOLLINS DW GODFREY CRA
Citation
Je. Baldwin et al., THE STEREOSPECIFIC SYNTHESIS OF (2S,3R) 3-CARBOXYPROLINE AND (2S,3R) 3-AMINOPROLINE, Tetrahedron, 51(17), 1995, pp. 5169-5180
Citations number
29
Categorie Soggetti
Chemistry Inorganic & Nuclear
Journal title
Tetrahedron → ACNP
ISSN journal
00404020
Volume
51
Issue
17
Year of publication
1995
Pages
5169 - 5180
Database
ISI
SICI code
0040-4020(1995)51:17<5169:TSSO(3>2.0.ZU;2-K
Abstract
Stereospecific syntheses of (2S,3R) 3-carboxyproline and (2S,3R) 3-ami noproline are reported which make use of the stereospecific alkylation of (4S)-N-(t-butyldimethylsilyl)azetidin-2-one 4-carboxylic acid with the cyclic sulfate derived from ethylene glycol.