INHIBITION OF HUMAN ERYTHROCYTE CALPAIN-I BY NOVEL QUINOLINE CARBOXAMIDES

Authors
GRAYBILL TL DOLLE RE OSIFO IK SCHMIDT SJ GREGORY JS HARRIS AL MILLER MS
Citation
Tl. Graybill et al., INHIBITION OF HUMAN ERYTHROCYTE CALPAIN-I BY NOVEL QUINOLINE CARBOXAMIDES, Bioorganic & medicinal chemistry letters, 5(4), 1995, pp. 387-392
Citations number
22
Categorie Soggetti
Chemistry Inorganic & Nuclear","Chemistry Medicinal
Journal title
Bioorganic & medicinal chemistry letters → ACNP
ISSN journal
0960894X
Volume
5
Issue
4
Year of publication
1995
Pages
387 - 392
Database
ISI
SICI code
0960-894X(1995)5:4<387:IOHECB>2.0.ZU;2-S
Abstract
1,4-Dihydro-4-oxo-3-quinolinecarboxamides are a class of non-peptide r eversible inhibitor of human erythrocyte Calpain I. The preparation an d in vitro evaluation of these compounds are discussed.