NOVEL ANALOGS OF TIAZOFURIN BY LAWESSON REAGENT EFFECTED CYCLIZATION

Citation
B. Golankiewicz et P. Januszczyk, NOVEL ANALOGS OF TIAZOFURIN BY LAWESSON REAGENT EFFECTED CYCLIZATION, Nucleosides & nucleotides, 14(3-5), 1995, pp. 313-316
Citations number
11
Categorie Soggetti
Biology
Journal title
ISSN journal
07328311
Volume
14
Issue
3-5
Year of publication
1995
Pages
313 - 316
Database
ISI
SICI code
0732-8311(1995)14:3-5<313:NAOTBL>2.0.ZU;2-Q
Abstract
2-Benzylthiazole-4-carboxamide 4 and 5-(beta-D-ribofuranosylamino) thi azole-4-carboxamide 10 were synthesized from phenylacetylamino- and fo rmylamino cyanoacetic acid esters 1a and 1b,respectively. The ribosyla tion reaction leading to 10 gave rise also to its alpha anomer as a mi nor product.