Jp. Demers et al., SELECTIVE INHIBITORS OF PROTEIN-KINASE-C IN A MODEL OF GRAFT-VS-HOST DISEASE, Bioorganic & medicinal chemistry letters, 4(20), 1994, pp. 2451-2456
A series of 3-aryl-4-arylidene-5-isoxazolones were found to be active
as inhibitors of PKC, and in ex-vivo and in vivo models of graft-versu
s-host disease.