FIRST APPLICATION OF THE DAKIN-WEST REACTION TO FMOC CHEMISTRY - SYNTHESIS OF THE KETOMETHYLENE TRIPEPTIDE OC-N-ALPHA-ASP(TBU)-(R,S)TYR(TBU)PSI(CO-CH2)GLY-OH

Authors
CASIMIR JR TURETTA C ETTOUATI L PARIS J
Citation
Jr. Casimir et al., FIRST APPLICATION OF THE DAKIN-WEST REACTION TO FMOC CHEMISTRY - SYNTHESIS OF THE KETOMETHYLENE TRIPEPTIDE OC-N-ALPHA-ASP(TBU)-(R,S)TYR(TBU)PSI(CO-CH2)GLY-OH, Tetrahedron letters, 36(27), 1995, pp. 4797-4800
Citations number
21
Categorie Soggetti
Chemistry Inorganic & Nuclear
Journal title
Tetrahedron letters → ACNP
ISSN journal
00404039
Volume
36
Issue
27
Year of publication
1995
Pages
4797 - 4800
Database
ISI
SICI code
0040-4039(1995)36:27<4797:FAOTDR>2.0.ZU;2-6
Abstract
A practical synthesis of a tripeptide containing a ketomethylene isost ere, suitably protected far introduction in Fmoc SPPS, has been carrie d out for the first time in Fmoc chemistry by using a modified Dakin-W est reaction.