H. Jendralla et al., EFFICIENT, SIMPLE PROCEDURES FOR THE LARGE-SCALE PREPARATION OF BUILDING-BLOCKS FOR ANGIOTENSIN(II) RECEPTOR ANTAGONISTS, Liebigs Annalen, (7), 1995, pp. 1253-1257
The kg-scale syntheses of p-formylbenzeneboronic acid 3c and the biphe
nyl derivatives 4a, 4b, and 4c, building blocks for angiotensin (II) r
eceptor antagonists, are reported.