DESYMMETRISATION OF BICYCLIC, MESO-ANHYDRIDES BY PROLINE ESTERS

Citation
Ig. Jones et al., DESYMMETRISATION OF BICYCLIC, MESO-ANHYDRIDES BY PROLINE ESTERS, Tetrahedron letters, 38(5), 1997, pp. 889-892
Citations number
11
Categorie Soggetti
Chemistry Inorganic & Nuclear
Journal title
ISSN journal
00404039
Volume
38
Issue
5
Year of publication
1997
Pages
889 - 892
Database
ISI
SICI code
0040-4039(1997)38:5<889:DOBMBP>2.0.ZU;2-W
Abstract
The desymmetrisation of cyclopropane and cyclopentane derived bicyclic meso-anhydrides using proline esters provides a versatile approach to the synthesis of enantiomerically pure amido acids which can subseque ntly be converted into beta-amino acid containing peptide analogues. ( C) 1997, Elsevier Science Ltd.