SYNTHESIS OF NOVEL INTRANUCLEAR DIAZASTEROIDS

Authors
MELLOR JM MERRIMAN GD
Citation
Jm. Mellor et Gd. Merriman, SYNTHESIS OF NOVEL INTRANUCLEAR DIAZASTEROIDS, Steroids, 60(10), 1995, pp. 693-698
Citations number
19
Categorie Soggetti
Biology,"Endocrynology & Metabolism
Journal title
Steroids → ACNP
ISSN journal
0039128X
Volume
60
Issue
10
Year of publication
1995
Pages
693 - 698
Database
ISI
SICI code
0039-128X(1995)60:10<693:SONID>2.0.ZU;2-Z
Abstract
By use of the aza Diels-Alder reaction a series of aminoisoquinolines and aminoquinolines have been elaborated to provide an effective synth esis of diverse diazasteroids. In particular, representative 1,11-diaz a-, 3,11-diaza-, and 4,11-diazasteroids have been synthesized from cyc lopentadiene. From dihydropyran a 4,11-diaza-15-oxa-D-homosteroid has been obtained.