THE CHEMISTRY OF INDOLES .66. A SYNTHESIS METHOD OF INDOLE-3-METHANAMINE AND OR GRAMINE FROM INDOLE-3-CARBOXALDEHYDE, AND ITS APPLICATION FOR THE SYNTHESIS OF BRASSININ, ITS 4-SUBSTITUTED ANALOGS, AND 1,3,4,5-TETRAHYDROPYRROLO[4,3,2-DE]QUINOLINE/

Authors
YAMADA F KOBAYASHI K SHIMIZU A AOKI N SOMEI M
Citation
F. Yamada et al., THE CHEMISTRY OF INDOLES .66. A SYNTHESIS METHOD OF INDOLE-3-METHANAMINE AND OR GRAMINE FROM INDOLE-3-CARBOXALDEHYDE, AND ITS APPLICATION FOR THE SYNTHESIS OF BRASSININ, ITS 4-SUBSTITUTED ANALOGS, AND 1,3,4,5-TETRAHYDROPYRROLO[4,3,2-DE]QUINOLINE/, Heterocycles, 36(12), 1993, pp. 2783-2804
Citations number
49
Categorie Soggetti
Chemistry Inorganic & Nuclear
Journal title
Heterocycles → ACNP
ISSN journal
03855414
Volume
36
Issue
12
Year of publication
1993
Pages
2783 - 2804
Database
ISI
SICI code
0385-5414(1993)36:12<2783:TCOI.A>2.0.ZU;2-L
Abstract
Simple conversion method of indole-3-carboxaldehyde into gramine and/o r indole-3-methanamine was developed. The present method realized shor t step syntheses of brassinin, 4-iodo-, methoxy-, 4-methoxy-, and 4-ni trobrassinin, 4-methoxyindole-3-acetonitrile, and 1, 3, 4, 5-tetrahydr opyrrolo[4, 3, 2-de]quinoline.