SYNTHESIS OF N-BENZYL-ACYLAMIDES AND N-HETEROARYLMETHYL-ACYLAMIDES BYREDUCTIVE N-ACYLATION OF ALDOXIMES WITH AMMONIUM FORMATE

Authors
BALICKI R KACZMAREK L
Citation
R. Balicki et L. Kaczmarek, SYNTHESIS OF N-BENZYL-ACYLAMIDES AND N-HETEROARYLMETHYL-ACYLAMIDES BYREDUCTIVE N-ACYLATION OF ALDOXIMES WITH AMMONIUM FORMATE, Gazzetta chimica italiana, 123(9), 1993, pp. 525-526
Citations number
23
Categorie Soggetti
Chemistry
Journal title
Gazzetta chimica italiana → ACNP
ISSN journal
00165603
Volume
123
Issue
9
Year of publication
1993
Pages
525 - 526
Database
ISI
SICI code
0016-5603(1993)123:9<525:SONANB>2.0.ZU;2-#
Abstract
Various (hetero)aryl aldoximes have been efficiently transformed to th e corresponding acylamides via reductive N-acylation, catalyzed by 10% palladium on carbon in the presence of ammonium formate as the hydrog en source in an alkanoic acid.