A REDUCTIVE AMINATION LACTAMIZATION PROCEDURE USING BOROHYDRIDE REAGENTS/

Authors
ABDELMAGID AF HARRIS BD MARYANOFF CA
Citation
Af. Abdelmagid et al., A REDUCTIVE AMINATION LACTAMIZATION PROCEDURE USING BOROHYDRIDE REAGENTS/, Synlett, (1), 1994, pp. 81-83
Citations number
15
Categorie Soggetti
Chemistry Inorganic & Nuclear
Journal title
Synlett → ACNP
ISSN journal
09365214
Issue
1
Year of publication
1994
Pages
81 - 83
Database
ISI
SICI code
0936-5214(1994):1<81:ARALPU>2.0.ZU;2-Z
Abstract
We report a procedure for tandem reductive amination-lactamization of aldehydes or ketones with aminoesters or ketoesters with primary amine s under mild conditions (NaBH(OAc)(3)/1,2-dichloroethane or NaBH4/MeOH ).