PREPARATION OF OPTICALLY-ACTIVE 6-SUBSTITUTED 2-PIPERIDONES BY OXIDATION OF THE CORRESPONDING OXAZOLOPIPERIDINES

Authors
LIENARD P VAREA T QUIRION JC HUSSON HP
Citation
P. Lienard et al., PREPARATION OF OPTICALLY-ACTIVE 6-SUBSTITUTED 2-PIPERIDONES BY OXIDATION OF THE CORRESPONDING OXAZOLOPIPERIDINES, Synlett, (2), 1994, pp. 143-144
Citations number
11
Categorie Soggetti
Chemistry Inorganic & Nuclear
Journal title
Synlett → ACNP
ISSN journal
09365214
Issue
2
Year of publication
1994
Pages
143 - 144
Database
ISI
SICI code
0936-5214(1994):2<143:POO62B>2.0.ZU;2-B
Abstract
Optically active 6-substituted 2-piperidones 4 and 5 were prepared in good yields (52%-80%) by treatment of corresponding aminoethers 2 and 3 with bromine in CHCl3.