ELECTROPHILIC FLUORINATION IN THE SYNTHESIS OF NEW FLUOROINDOLES

Authors
HODSON HF MADGE DJ SLAWIN ANZ WIDDOWSON DA WILLIAMS DJ
Citation
Hf. Hodson et al., ELECTROPHILIC FLUORINATION IN THE SYNTHESIS OF NEW FLUOROINDOLES, Tetrahedron, 50(6), 1994, pp. 1899-1906
Citations number
25
Categorie Soggetti
Chemistry Inorganic & Nuclear
Journal title
Tetrahedron → ACNP
ISSN journal
00404020
Volume
50
Issue
6
Year of publication
1994
Pages
1899 - 1906
Database
ISI
SICI code
0040-4020(1994)50:6<1899:EFITSO>2.0.ZU;2-1
Abstract
Fluorination of trialkylstannylindoles with caesium fluoroxysulfate or Selectfluor(TM) was investigated for the synthesis of inter-alia 2- a nd 3-fluoroindoles. Caseium fluoroxysulfate gave good yields of these potentially useful intermediates; Selectfluor provided lower yields.