2 NEW PROCEDURES FOR THE INTRODUCTION OF BENZYL-TYPE PROTECTING GROUPS FOR THIOLS

Authors
RICHTER LS MARSTERS JC GADEK TR
Citation
Ls. Richter et al., 2 NEW PROCEDURES FOR THE INTRODUCTION OF BENZYL-TYPE PROTECTING GROUPS FOR THIOLS, Tetrahedron letters, 35(11), 1994, pp. 1631-1634
Citations number
12
Categorie Soggetti
Chemistry Inorganic & Nuclear
Journal title
Tetrahedron letters → ACNP
ISSN journal
00404039
Volume
35
Issue
11
Year of publication
1994
Pages
1631 - 1634
Database
ISI
SICI code
0040-4039(1994)35:11<1631:2NPFTI>2.0.ZU;2-F
Abstract
Two new methods for the benzylation of thiols are described: a) direct S-alkylation with para-substituted benzylic cations; and b) reductive S-alkylations of 2-aminothiols. Both methods provide efficient routes for the introduction of benzyl-type protecting groups in high yields.