D. Achard et al., PERHYDROTHIOPYRANOPYRROLES DERIVATIVES - A NOVEL SERIES OF POTENT ANDSELECTIVE NONPEPTIDE NK1 ANTAGONISTS, Bioorganic & medicinal chemistry letters, 4(5), 1994, pp. 669-672
The synthesis of RP 73467, a representative of 4,4-diphenyl perhydroth
iopyrano[2,3-c]-pyrroles 1-oxides, a new sefies of potent and selectiv
e nonpeptide NKI Substance P antagonists, is descfibed.