EFFICIENT SYNTHESIS OF 3-SUBSTITUTED INDOLES BY PALLADIUM-CATALYZED COUPLING REACTION OF 3-TRIBUTYLSTANNYLINDOLES WITH ORGANIC TRIFLATES AND HALIDES

Authors
CIATTINI PG MORERA E ORTAR G
Citation
Pg. Ciattini et al., EFFICIENT SYNTHESIS OF 3-SUBSTITUTED INDOLES BY PALLADIUM-CATALYZED COUPLING REACTION OF 3-TRIBUTYLSTANNYLINDOLES WITH ORGANIC TRIFLATES AND HALIDES, Tetrahedron letters, 35(15), 1994, pp. 2405-2408
Citations number
24
Categorie Soggetti
Chemistry Inorganic & Nuclear
Journal title
Tetrahedron letters → ACNP
ISSN journal
00404039
Volume
35
Issue
15
Year of publication
1994
Pages
2405 - 2408
Database
ISI
SICI code
0040-4039(1994)35:15<2405:ESO3IB>2.0.ZU;2-C
Abstract
The palladium-catalyzed reaction of 1-tosyl-3-tributylstannylindoles 2 with a variety of vinyl, aryl, and heteroaryl triflates and halides ( 1) provides a general and efficient method for the synthesis of 3-subs tituted indoles 3.