A FACILE ONE-POT SYNTHESIS OF PYRAZOLOTHIAZOLES

Authors
Citation
Vr. Rao et Tvp. Rao, A FACILE ONE-POT SYNTHESIS OF PYRAZOLOTHIAZOLES, Indian journal of chemistry. Sect. B: organic chemistry, including medical chemistry, 33(5), 1994, pp. 470-473
Citations number
10
Categorie Soggetti
Chemistry Inorganic & Nuclear
ISSN journal
03764699
Volume
33
Issue
5
Year of publication
1994
Pages
470 - 473
Database
ISI
SICI code
0376-4699(1994)33:5<470:AFOSOP>2.0.ZU;2-V
Abstract
A one-pot synthesis of 3-[2-(3, 4, 5-trisubstituted-1H-pyrazol-1-yl) - 4-thiazolyl] -2H-1-benzopyran-2-ones (3) has been carried out by conde nsation of 3,4,5-tri-substituted-1-thiocarbamoylpyrazoles (1) with sub stituted 3-acetylcoumarins(2)in the presence of I2 or Br2 in dioxane a nd DMF on a steam-bath.