Ec. Taylor et Je. Dowling, SYNTHESIS OF A PYRIMIDO[4,5-B]AZEPINE ANALOG OF 5,10-DIDEAZA-5,6,7,8-TETRAHYDROFOLIC ACID (DDATHF), Bioorganic & medicinal chemistry letters, 7(4), 1997, pp. 453-456
The synthesis and biological evaluation of a pyrimido[4,5-b]azepine-ba
sed analog of DDATHF, a potential chemotherapeutic agent, are describe
d. (C) 1997, Elsevier Science Ltd.