SELECTIVE AZIRIDINATION OF OLEFINIC ESTERS

Authors
DESHMUKH M CHAVAN P KHARADE D
Citation
M. Deshmukh et al., SELECTIVE AZIRIDINATION OF OLEFINIC ESTERS, Monatshefte fuer Chemie, 125(6-7), 1994, pp. 743-746
Citations number
14
Categorie Soggetti
Chemistry
Journal title
Monatshefte fuer Chemie → ACNP
ISSN journal
00269247
Volume
125
Issue
6-7
Year of publication
1994
Pages
743 - 746
Database
ISI
SICI code
0026-9247(1994)125:6-7<743:SAOOE>2.0.ZU;2-P
Abstract
Oxidation of 3-amino-2-isobutylquinazoline-4-one (2) with lead tetraac etate at -20-degrees-C gave N-acetoxyamino-2-isobutylquinazolin-4-one (3), which selectively aziridinated olefinic esters to yield substitut ed lquinazolin-4'-one-3'-yl)-aziridine-2-carboxylates 5a-q.