TMSO-TRIFLATE-ASSISTED ADDITION OF ENOLS TO HETEROAROMATIC IMINES OR HYDROXYAMINAL INTERMEDIATES

Authors
MOUTOU JL SCHMITT M WERMUTH CG BOURGUIGNON JJ
Citation
Jl. Moutou et al., TMSO-TRIFLATE-ASSISTED ADDITION OF ENOLS TO HETEROAROMATIC IMINES OR HYDROXYAMINAL INTERMEDIATES, Tetrahedron letters, 35(37), 1994, pp. 6883-6886
Citations number
10
Categorie Soggetti
Chemistry Inorganic & Nuclear
Journal title
Tetrahedron letters → ACNP
ISSN journal
00404039
Volume
35
Issue
37
Year of publication
1994
Pages
6883 - 6886
Database
ISI
SICI code
0040-4039(1994)35:37<6883:TAOETH>2.0.ZU;2-H
Abstract
TMSOTf-promoted reaction of heteroaromatic imines or hydroxyaminal int ermediates with various enolic ketones are reported. This reaction con stitutes an original and regioselective mode of alkylation of exocycli c amines of heterocyclic amidines.