A NOVEL ONE-POT CONVERSION OF METHYL SULFONES TO SULFONAMIDES

Authors
HUANG HC REINHARD EJ REITZ DB
Citation
Hc. Huang et al., A NOVEL ONE-POT CONVERSION OF METHYL SULFONES TO SULFONAMIDES, Tetrahedron letters, 35(39), 1994, pp. 7201-7204
Citations number
13
Categorie Soggetti
Chemistry Inorganic & Nuclear
Journal title
Tetrahedron letters → ACNP
ISSN journal
00404039
Volume
35
Issue
39
Year of publication
1994
Pages
7201 - 7204
Database
ISI
SICI code
0040-4039(1994)35:39<7201:ANOCOM>2.0.ZU;2-G
Abstract
A one-pot synthesis of sulfonamides from methyl sulfones has been deve loped. Treatment of methyl sulfones with base and trialkylboranes gave the corresponding rearranged sulfinic acid salts which were converted to sulfonamides during oxidative-amination workup.