THE SYNTHESIS OF AZATRYPTOPHANE DERIVATIVES

Authors
SVETE J STANOVNIK B TISLER M
Citation
J. Svete et al., THE SYNTHESIS OF AZATRYPTOPHANE DERIVATIVES, Journal of heterocyclic chemistry, 31(5), 1994, pp. 1259-1266
Citations number
8
Categorie Soggetti
Chemistry Inorganic & Nuclear
Journal title
Journal of heterocyclic chemistry → ACNP
ISSN journal
0022152X
Volume
31
Issue
5
Year of publication
1994
Pages
1259 - 1266
Database
ISI
SICI code
0022-152X(1994)31:5<1259:TSOAD>2.0.ZU;2-2
Abstract
Optically active and racemic isomers of aspartic acid (1) were transfo rmed into the corresponding N-trifluoroacetyl-5-bromo-4-oxonorvaline m ethyl esters (6, R = Me) and N-trifluoroacetyl-3-formylalanine methyl esters 13, which were used as starting compounds in the synthesis of b eta-heteroaryl substituted-alpha-amino acids.