D. Hill et al., SYNTHESIS OF A POTENT AND SELECTIVE NONPEPTIDE CCK-B GASTRIN RECEPTORANTAGONIST TRITIATED LIGAND, Bioorganic & medicinal chemistry letters, 3(5), 1993, pp. 885-888
The synthesis of a novel, potent and selective non-peptide gastrin/CCK
-B receptor antagonist in a tritiated form is described, via a route w
hich allows for introduction of the radiolabel in the final step.