SYNTHESIS OF (1R,4R,7S) AND NYLMETHYL-7-METHYL-2,5-DIAZABICYCLO[2.2.1]HEPTANES VIA REGIOSELECTIVE OPENING OF 3,4-EPOXY-D-PROLINE WITH LITHIUM DIMETHYL CUPRATE

Authors
REMUZON P BOUZARD D CLEMENCIN C DUSSY C ESSIZ M JACQUET JP SAINTGERMAIN J
Citation
P. Remuzon et al., SYNTHESIS OF (1R,4R,7S) AND NYLMETHYL-7-METHYL-2,5-DIAZABICYCLO[2.2.1]HEPTANES VIA REGIOSELECTIVE OPENING OF 3,4-EPOXY-D-PROLINE WITH LITHIUM DIMETHYL CUPRATE, Journal of heterocyclic chemistry, 30(2), 1993, pp. 517-523
Citations number
13
Categorie Soggetti
Chemistry Inorganic & Nuclear
Journal title
Journal of heterocyclic chemistry → ACNP
ISSN journal
0022152X
Volume
30
Issue
2
Year of publication
1993
Pages
517 - 523
Database
ISI
SICI code
0022-152X(1993)30:2<517:SO(AN>2.0.ZU;2-Y
Abstract
The synthesis of (1S, 1S, 7S)- and (IR, 4R, ylmethyl-7-methyl-2,5-diaz abicyclo-[2.2.1]heptanes (20) and (22) from trans 4-hydroxy-L-proline is described.