SOLID-PHASE SYNTHESIS OF PHOSPHINIC PEPTIDES

Authors
CAMPAGNE JM COSTE J GUILLOU L HEITZ A JOUIN P
Citation
Jm. Campagne et al., SOLID-PHASE SYNTHESIS OF PHOSPHINIC PEPTIDES, Tetrahedron letters, 34(26), 1993, pp. 4181-4184
Citations number
15
Categorie Soggetti
Chemistry Inorganic & Nuclear
Journal title
Tetrahedron letters → ACNP
ISSN journal
00404039
Volume
34
Issue
26
Year of publication
1993
Pages
4181 - 4184
Database
ISI
SICI code
0040-4039(1993)34:26<4181:SSOPP>2.0.ZU;2-G
Abstract
The absence of a coupling reaction between a phosphinic acid and an am ino ester during activation with the reagents BOP or PyBOP allowed the synthesis of phosphinopeptides from phospho-analogues of dipeptides, unprotected on the phosphinic acid.