A NOVEL ONE-POT SYNTHESIS OF SUBSTITUTED 5-BENZOYL-1H,6H-PYRANO[2,3-C]PYRAZOLONE AND 5-ACETYLAMINO-1H, 6H-PYRANO[2,3-C]PYRAZOLONE

Citation
Vk. Ahluwalia et al., A NOVEL ONE-POT SYNTHESIS OF SUBSTITUTED 5-BENZOYL-1H,6H-PYRANO[2,3-C]PYRAZOLONE AND 5-ACETYLAMINO-1H, 6H-PYRANO[2,3-C]PYRAZOLONE, Indian journal of chemistry. Sect. B: organic chemistry, including medical chemistry, 32(9), 1993, pp. 960-962
Citations number
12
Categorie Soggetti
Chemistry Inorganic & Nuclear
ISSN journal
03764699
Volume
32
Issue
9
Year of publication
1993
Pages
960 - 962
Database
ISI
SICI code
0376-4699(1993)32:9<960:ANOSOS>2.0.ZU;2-X
Abstract
A convenient one-pot synthesis of some 5-benzoyl- and 5-acetylamino-1H , 6H-pyrano[2, 3-c]pyrazolones (4) by the reaction of 2-pyrazolin-5-on es (1) with hippuric/aceturic acid and triethyl orthoformate in the pr esence of acetic anhydride, in good yield (75-85%) has been described.