AN EFFICIENT SYNTHESIS OF NEW PHENYLPYRROLIZINE AND PHENYLPYRROLOPYRAZINE DERIVATIVES

Authors
TEMBO ON DALLEMAGNE P RAULT S ROBBA M
Citation
On. Tembo et al., AN EFFICIENT SYNTHESIS OF NEW PHENYLPYRROLIZINE AND PHENYLPYRROLOPYRAZINE DERIVATIVES, Heterocycles, 36(9), 1993, pp. 2129-2137
Citations number
6
Categorie Soggetti
Chemistry Inorganic & Nuclear
Journal title
Heterocycles → ACNP
ISSN journal
03855414
Volume
36
Issue
9
Year of publication
1993
Pages
2129 - 2137
Database
ISI
SICI code
0385-5414(1993)36:9<2129:AESONP>2.0.ZU;2-9
Abstract
Synthesis of new 3-phenyl-2,3-dihydro-1H-pyrrolizine derivatives is ac hieved starting from 3-amino-3-phenylpropionic acid via an iminium sal t. The reactivity of this system is studied and the new nyl-1,2,3,4-te trahydropyrrolo-[1,2-a]pyrazin-1-one derivatives are synthesized, via a Beckmann's rearrangment.