INTRAMOLECULAR TRANSAMINATIONS OF ENAMINONES - A SYNTHESIS OF FUSED, POLYCYCLIC, N-ARYL PYRIDONES

Authors
FRIARY RJ SEIDL V SCHWERDT JH COHEN MP HOU D NAFISSI M
Citation
Rj. Friary et al., INTRAMOLECULAR TRANSAMINATIONS OF ENAMINONES - A SYNTHESIS OF FUSED, POLYCYCLIC, N-ARYL PYRIDONES, Tetrahedron, 49(33), 1993, pp. 7169-7178
Citations number
21
Categorie Soggetti
Chemistry Inorganic & Nuclear
Journal title
Tetrahedron → ACNP
ISSN journal
00404020
Volume
49
Issue
33
Year of publication
1993
Pages
7169 - 7178
Database
ISI
SICI code
0040-4020(1993)49:33<7169:ITOE-A>2.0.ZU;2-9
Abstract
2-Arylamino-3-pyridinecarbonyl chlorides acylated the beta-carbon atom s of enamines, and the resulting enaminones cyclized to give a series of fused polycyclic N-aryl pyridones. The series included 9,10-tetrahy drobenzo[b][1,8]naphthyridin-5(7H)-one (Sch 40120), an antipsoriatic a gent.