A. Benarab et G. Guillaumet, SYNTHESIS AND SEROTONERGIC ACTIVITY OF METHYLAMINO)BUTYL]-8-AZASPIRO[4.5]DECANE-7,9-DIONE, Heterocycles, 36(10), 1993, pp. 2327-2333
The synthesis of compound (9), a nitrogen-containing bioisostere of th
e 1,4-benzodioxane moiety of the MDL 72832, is detailed. This compound
showed a moderate affinity for the 5-HT1A receptors.