A palladium-catalyzed domino process to 1-benzazepines

Authors
Dyker, G Markwitz, H
Citation
G. Dyker et H. Markwitz, A palladium-catalyzed domino process to 1-benzazepines, SYNTHESIS-S, (12), 1998, pp. 1750-1754
Citations number
14
Categorie Soggetti
Chemistry & Analysis","Organic Chemistry/Polymer Science
Journal title
SYNTHESIS-STUTTGART
ISSN journal
00397881 → ACNP
Issue
12
Year of publication
1998
Pages
1750 - 1754
Database
ISI
SICI code
0039-7881(199812):12<1750:APDPT1>2.0.ZU;2-7
Abstract
2-Iodonailine (1) undergoes a palladium-catalyzed annulation reaction with homoallylic alcohols 2 leading to 1-benzazepines 4. This domino process is the result of a Heck reaction with double bond migration followed by cycloc ondensation.