Synthesis of diacylamines and the preparation of alpha-amino-acylureas, a new type of alpha-amino acid derivatives

Citation
I. Weisz et al., Synthesis of diacylamines and the preparation of alpha-amino-acylureas, a new type of alpha-amino acid derivatives, BIOORG MED, 8(22), 1998, pp. 3241-3244
Citations number
15
Categorie Soggetti
Chemistry & Analysis
Journal title
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
ISSN journal
0960894X → ACNP
Volume
8
Issue
22
Year of publication
1998
Pages
3241 - 3244
Database
ISI
SICI code
0960-894X(19981117)8:22<3241:SODATP>2.0.ZU;2-X
Abstract
Sixteen new and one known unsymmetrical open-chain diacylamines were synthe sized by sodium methoxide catalyzed acylation of amides with carboxylic est ers and acylamino-carboxylic esters, or acylureas with acylamino-carboxylic esters and alpha-amino acid esters. (C) 1998 Elsevier Science Ltd. All rig hts reserved.