Aminoacrylates. II. An efficient synthesis of alpha-pyridones by heterocyclic annelation reactions of magnesium amides derived from sec-aminoacrylates with methyl propiolate

Authors
Koike, T Takeuchi, N Tobinaga, S
Citation
T. Koike et al., Aminoacrylates. II. An efficient synthesis of alpha-pyridones by heterocyclic annelation reactions of magnesium amides derived from sec-aminoacrylates with methyl propiolate, CHEM PHARM, 47(1), 1999, pp. 128-130
Citations number
17
Categorie Soggetti
Chemistry & Analysis
Journal title
CHEMICAL & PHARMACEUTICAL BULLETIN
ISSN journal
00092363 → ACNP
Volume
47
Issue
1
Year of publication
1999
Pages
128 - 130
Database
ISI
SICI code
0009-2363(199901)47:1<128:AIAESO>2.0.ZU;2-N
Abstract
The reactions of magnesium amides 4 derived from sec-aminoacrylates 3 and e thylmagnesium bromide with methyl propiolate (2) afforded alpha-pyridones. This provides an efficient heterocyclic annelation reaction.