A solid-phase synthesis of functionalized 6-, 7- and 8-membered azacycles via olefin metathesis

Authors
Pernerstorfer, J Schuster, M Blechert, S
Citation
J. Pernerstorfer et al., A solid-phase synthesis of functionalized 6-, 7- and 8-membered azacycles via olefin metathesis, SYNTHESIS-S, (1), 1999, pp. 138-144
Citations number
28
Categorie Soggetti
Chemistry & Analysis","Organic Chemistry/Polymer Science
Journal title
SYNTHESIS-STUTTGART
ISSN journal
00397881 → ACNP
Issue
1
Year of publication
1999
Pages
138 - 144
Database
ISI
SICI code
0039-7881(199901):1<138:ASSOF6>2.0.ZU;2-1
Abstract
A modular solid-phase synthesis of functionalized aza-cycles is described. The approach is based on a ring-closing metathesis to form heterocycles of different ring sizes. Furthermore, the epoxidation of the primarily formed cyclic double bond has been investigated.