5-chloro-N-(4-methoxy-3-piperazin-1-yl-phenyl)-3-methyl-2-benzothiophenesulfonamide (SB-271046): A potent, selective, and orally bioavailable 5-HT6 receptor antagonist

Bromidge, SM Brown, AM Clarke, SE Dodgson, K Gager, T Grassam, HL Jeffrey, PM Joiner, GF King, FD Middlemiss, DN Moss, SF Newman, H Riley, G Routledge, C Wyman, P

Sm. Bromidge et al., 5-chloro-N-(4-methoxy-3-piperazin-1-yl-phenyl)-3-methyl-2-benzothiophenesulfonamide (SB-271046): A potent, selective, and orally bioavailable 5-HT6 receptor antagonist, J MED CHEM, 42(2), 1999, pp. 202-205

16

Chemistry & Analysis

JOURNAL OF MEDICINAL CHEMISTRY

00222623 → ACNP

42

2

1999

202 - 205

ISI

0022-2623(19990128)42:2<202:5>2.0.ZU;2-R