DOCETAXEL (TAXOTERE) DERIVATIVES - NOVEL NBCL3-BASED STEREOSELECTIVE APPROACH TO 2'-METHYLDOCETAXEL

Authors
DENIS JN FKYERAT A GIMBERT Y COUTTEREZ C MANTELLIER P JOST S GREENE AE
Citation
Jn. Denis et al., DOCETAXEL (TAXOTERE) DERIVATIVES - NOVEL NBCL3-BASED STEREOSELECTIVE APPROACH TO 2'-METHYLDOCETAXEL, Journal of the Chemical Society. Perkin transactions. I, (14), 1995, pp. 1811-1815
Citations number
30
Categorie Soggetti
Chemistry Inorganic & Nuclear
Journal title
Journal of the Chemical Society. Perkin transactions. I → ACNP
ISSN journal
0300922X
Issue
14
Year of publication
1995
Pages
1811 - 1815
Database
ISI
SICI code
0300-922X(1995):14<1811:D(D-NN>2.0.ZU;2-G
Abstract
The C-2 methylated 2S,3R and 2R,3S side chains of docetaxel have been enantioselectively prepared and esterified with protected 10-deacetylb accatin III to provide novel analogues of docetaxel.