SYNTHESIS OF SOME NEW PYRROLO HETEROCYCLES - CONDENSATION OF 4-CARBOMETHOXY-1-METHYL-2,3-DIOXOPYRROLIDINE WITH PRIMARY AMINES

Authors
Citation
Ma. Sofan, SYNTHESIS OF SOME NEW PYRROLO HETEROCYCLES - CONDENSATION OF 4-CARBOMETHOXY-1-METHYL-2,3-DIOXOPYRROLIDINE WITH PRIMARY AMINES, Die Pharmazie, 52(4), 1997, pp. 276-278
Citations number
23
Categorie Soggetti
Pharmacology & Pharmacy",Chemistry
Journal title
ISSN journal
00317144
Volume
52
Issue
4
Year of publication
1997
Pages
276 - 278
Database
ISI
SICI code
0031-7144(1997)52:4<276:SOSNPH>2.0.ZU;2-A
Abstract
2,3-Dioxypyrrolidine (1) was prepared and treated with primary aromati c amines to give the 4-carbamoyl derivatives 2a-d which cyclized to py rrolo[3,4-c]quinolines 3a, b and 4. Condensation of 1 with aminoazoles gave che linearly fused pyrroloheterocycles 5-7. The triazinopyrrole ring system 9 was obtained from 8 and thiosemicarbazide.