A FACILE COPPER-CATALYZED ULLMANN CONDENSATION - N-ARYLATION OF HETEROCYCLIC-COMPOUNDS CONTAINING AN -NHCO- MOIETY

Citation
M. Sugahara et T. Ukita, A FACILE COPPER-CATALYZED ULLMANN CONDENSATION - N-ARYLATION OF HETEROCYCLIC-COMPOUNDS CONTAINING AN -NHCO- MOIETY, Chemical and Pharmaceutical Bulletin, 45(4), 1997, pp. 719-721
Citations number
18
Categorie Soggetti
Pharmacology & Pharmacy",Chemistry
ISSN journal
00092363
Volume
45
Issue
4
Year of publication
1997
Pages
719 - 721
Database
ISI
SICI code
0009-2363(1997)45:4<719:AFCUC->2.0.ZU;2-3
Abstract
N-Aryl heterocyclic compounds were synthesized from aryl halides and h eterocyclic compounds containing an -NHCO- moiety by using a catalytic amount (1-10 mol%) of a commercially available copper catalyst in sat isfactory yields. This catalytic reaction was applicable to the synthe sis of N-aryl-2-pyridone, -2-pyrrolidone,-1(2H)-isoquinolone, -1(2H)-p hthalazinone, -4(3H)-quinazolinone and -1,2,3-benzotriazin-4(3H)-one d erivatives.