Us. Pathak et al., SYNTHESIS OF NOVEL HIENO[2,3-D][1,2,4]TRIAZOLO[1,5-A]PYRIMIDIN-5-ONES, Indian journal of chemistry. Sect. B: organic chemistry, including medical chemistry, 36(7), 1997, pp. 566-571
A facile and simple synthesis for ,2,3,4-tetrahydrothieno[2,3-6]-pyrim
idin-4(3H)-one 3a is described and from this precursor, a series of hi
therto unreported linear ,2-disubstituted-6,-dimethyl-[1H,5H]-thieno[2
,3-d] [1,2,4]triazolo[1,5-a]pyrimidin-5-ones 6a-0 have been synthesise
d by the cyclocondensation of the corresponding mino-5,6-dimethylthien
o[2,3-d]pyrimidin-4(3H)-ones 5a,b with various one carbon donors.