NOVEL AND CONVENIENT SYNTHESIS OF 1,4-DIHYDROPYRIDAZINES AND PYRIDAZINES FROM AMINOCARBONYLAZOALKENES

Authors
ATTANASI OA FILIPPONE P FIORUCCI C MANTELLINI F
Citation
Oa. Attanasi et al., NOVEL AND CONVENIENT SYNTHESIS OF 1,4-DIHYDROPYRIDAZINES AND PYRIDAZINES FROM AMINOCARBONYLAZOALKENES, Synlett, (12), 1997, pp. 1361-1362
Citations number
40
Journal title
Synlett → ACNP
ISSN journal
09365214
Issue
12
Year of publication
1997
Pages
1361 - 1362
Database
ISI
SICI code
0936-5214(1997):12<1361:NACSO1>2.0.ZU;2-L
Abstract
1-Unsubstituted 1,4-dihydropyridazines have been obtained in good to e xcellent yields by reaction of aminocarbonylazoalkenes with beta-trica rbonyl compounds under mild conditions. Treatment at room temperature of 1-unsubstituted 1,4-dihydropyridazines with phenyltrimethylammonium tribromide directly afforded the relevant pyridazine derivatives in h igh yield.