AN EFFICIENT SYNTHESIS OF 4-ARYL AND 4-VINYLPHENYLALANINES BY STILLE CROSS-COUPLING REACTION

Authors
MORERA E ORTAR G
Citation
E. Morera et G. Ortar, AN EFFICIENT SYNTHESIS OF 4-ARYL AND 4-VINYLPHENYLALANINES BY STILLE CROSS-COUPLING REACTION, Synlett, (12), 1997, pp. 1403-1405
Citations number
27
Journal title
Synlett → ACNP
ISSN journal
09365214
Issue
12
Year of publication
1997
Pages
1403 - 1405
Database
ISI
SICI code
0936-5214(1997):12<1403:AESO4A>2.0.ZU;2-Q
Abstract
The palladium-catalyzed reaction of N-Boc-4-trimethylstannyl-L-phenyla lanine methyl ester (1) with a variety of aryl and vinyl iodides and t riflates (2) affords the corresponding 4-aryl and 4-vinylphenylalanine s 3 in synthetically useful yields.