AMINOLYSIS OF N-TRITYLAMINO ACID BENZOTRIAZOLYL ESTERS WITH CONCENTRATED AQUEOUS AMINES AND ITS APPLICATIONS IN SYNTHESIS

Authors
MAMOS P DALATSIS E ATHANASSOPOULOS C BALAYIANNIS G PAPAIOANNOU D FRANCIS GW
Citation
P. Mamos et al., AMINOLYSIS OF N-TRITYLAMINO ACID BENZOTRIAZOLYL ESTERS WITH CONCENTRATED AQUEOUS AMINES AND ITS APPLICATIONS IN SYNTHESIS, Acta chemica Scandinavica, 52(2), 1998, pp. 227-231
Citations number
6
Categorie Soggetti
Chemistry,Biology
Journal title
Acta chemica Scandinavica → ACNP
ISSN journal
0904213X
Volume
52
Issue
2
Year of publication
1998
Pages
227 - 231
Database
ISI
SICI code
0904-213X(1998)52:2<227:AONABE>2.0.ZU;2-R
Abstract
Aminolysis of (S)-N-tritylamino acid benzotriazolyl eaters with concen trated aqueous amines produces high yields of the corresponding amides which can be readily detritylated with p-toluensulfonic acid or reduc ed with lithium aluminium hydride to provide chiral ethane-1;2-diamine derivatives.