A MILD METHOD FOR FORMYLATING AMINO ESTERS WITHOUT USING ANY FORMYLATING AGENT

Authors
GIARD T BENARD D PLAQUEVENT JC
Citation
T. Giard et al., A MILD METHOD FOR FORMYLATING AMINO ESTERS WITHOUT USING ANY FORMYLATING AGENT, Synthesis, (3), 1998, pp. 297-300
Citations number
21
Categorie Soggetti
Chemistry Inorganic & Nuclear
Journal title
Synthesis → ACNP
ISSN journal
00397881
Issue
3
Year of publication
1998
Pages
297 - 300
Database
ISI
SICI code
0039-7881(1998):3<297:AMMFFA>2.0.ZU;2-Q
Abstract
A simple and mild method for the N-formylation of alpha-amino esters i s described via an intermediate oxaziridine. This procedure avoids the necessity of specific formylating agents and yields the N-formyl spec ies in high yield and without racemization.