A CONVENIENT SYNTHESIS OF DIALKYL [2-(BROMOMETHYL)AZIRIDIN-1-YL]METHYL]PHOSPHONATES, NEW HETEROCYCLIC BETA-AZAPHOSPHONATES

Authors
STEVENS C VERBEKE A DEKIMPE N
Citation
C. Stevens et al., A CONVENIENT SYNTHESIS OF DIALKYL [2-(BROMOMETHYL)AZIRIDIN-1-YL]METHYL]PHOSPHONATES, NEW HETEROCYCLIC BETA-AZAPHOSPHONATES, Synlett, (2), 1998, pp. 180
Citations number
12
Categorie Soggetti
Chemistry Inorganic & Nuclear
Journal title
Synlett → ACNP
ISSN journal
09365214
Issue
2
Year of publication
1998
Database
ISI
SICI code
0936-5214(1998):2<180:ACSOD[>2.0.ZU;2-5
Abstract
Dialkyl [[2-(bromomethyl)aziridin-1-yl]methyl] phosphonates were prepa red in good yield by a convenient procedure involving the reaction of 1,3,5-triallylhexahydro[1,3,5]triazine with dialkyl phosphites, subseq uent bromination and final ring closure upon treatment with sodium bor ohydride in methanol.